α4β2烟碱乙酰胆碱受体的部分激动剂,TC 2559 (fumarate) is a CNS-selective partial agonist for α4β2 subunit-containing nicotinic acetylcholine receptors (nAChRs) with an EC50 value of 0.18 μM for calcium signaling in HEK293 cells expressing human recombinant nAChRs.
α4β2烟碱乙酰胆碱受体的部分激动剂,TC 2559 (fumarate) is a CNS-selective partial agonist for α4β2 subunit-containing nicotinic acetylcholine receptors (nAChRs) with an EC50 value of 0.18 μM for calcium signaling in HEK293 cells expressing human recombinant nAChRs.